Thursday, January 19, 2017

Covalent Modulators of the Vacuolar ATPase

Covalent Modulators of the Vacuolar ATPase

Ying-Chu Chen, Keriann M. Backus, Maria Merkulova, Christina Yang, Dennis Brown, Benjamin F. Cravatt, and Chao Zhang
J. Am. Chem. Soc., 2017, 139 (2), pp 639–642

Overcoming EGFR Resistance by Monovalent and Bident Inhibitors Targeting Cys775

  Zhengnian Li , Jie Jiang , Yaning Wang , Scott B. Ficarro , Stephen J. Collins , Tyler S. Beyett , Ilse K. Schaeffner , Isidoro Tavares , ...