Thursday, January 19, 2017

Covalent Modulators of the Vacuolar ATPase

Covalent Modulators of the Vacuolar ATPase

Ying-Chu Chen, Keriann M. Backus, Maria Merkulova, Christina Yang, Dennis Brown, Benjamin F. Cravatt, and Chao Zhang
J. Am. Chem. Soc., 2017, 139 (2), pp 639–642

Sulfonyl-Imidazopyridines Decouple Reactivity from Stability for Ligandability Mapping and Covalent Inhibitor Discovery

Zhihong Li , Madeleine L. Ware , Phillip W. Gingrich , Bissan Al-Lazikani , Ku-Lung Hsu;   Journal American Chemical Society (2026) 148 (39...