Thursday, March 2, 2017

Ligand and Target Discovery by Fragment-Based Screening in Human Cells

Christopher G. Parker, Andrea Galmozzi, Yujia Wang, Bruno E. Correia, Kenji Sasaki, Christopher M. Joslyn, Arthur S. Kim, Cullen L. Cavallaro, R. Michael Lawrence, Stephen R. Johnson, Iñigo Narvaiza, Enrique Saez, Enrique Saez,Enrique Saez, Benjamin F. Cravatt6, Benjamin F. Cravatt

DOI: 10.1016/j.cell.2016.12.029

Rational Design of CDK12/13 and BRD4 Molecular Glue Degraders

Nathanael Schiander Gray ,  Zhe Zhuang ,  Woong Sub Byun ,  Zuzanna Kozicka ,  Katherine Donovan ,  Brendan Dwyer ,  Abby Thornhill ,  Hanna...