Tuesday, September 2, 2025

Covalent chemical probes

Backus, K.M., Wilson, A.J. 

Commun Chem 8, 266 (2025). 

https://doi.org/10.1038/s42004-025-01652-6


Overcoming EGFR Resistance by Monovalent and Bident Inhibitors Targeting Cys775

  Zhengnian Li , Jie Jiang , Yaning Wang , Scott B. Ficarro , Stephen J. Collins , Tyler S. Beyett , Ilse K. Schaeffner , Isidoro Tavares , ...