Tuesday, September 2, 2025

Covalent chemical probes

Backus, K.M., Wilson, A.J. 

Commun Chem 8, 266 (2025). 

https://doi.org/10.1038/s42004-025-01652-6


Late-stage functionalization with strain-release warheads enables tunable covalent inhibition

Zachary P. Shultz, Ansar Lee-Sam, Yun-Pu Chang, Luxin Sun, Dylan Grassie, Alessio Gabellini, Kyle Pedretty, Thomas Scattolin, Victoria Izumi...